{"id":13642,"date":"2020-10-26T12:39:19","date_gmt":"2020-10-26T12:39:19","guid":{"rendered":"https:\/\/higeacbd.com\/huiles\/pharmacodynamique-et-pharmacocinetique\/"},"modified":"2021-11-12T11:23:57","modified_gmt":"2021-11-12T11:23:57","slug":"pharmacodynamique-et-pharmacocinetique","status":"publish","type":"post","link":"https:\/\/higeacbd.com\/fr\/datos\/pharmacodynamique-et-pharmacocinetique","title":{"rendered":"Pharmacodynamique et pharmacocin\u00e9tique"},"content":{"rendered":"<p>[et_pb_section fb_built=&#8221;1&#8243; admin_label=&#8221;Hero&#8221; _builder_version=&#8221;4.6.6&#8243; background_color=&#8221;rgba(255,255,255,0.65)&#8221; background_image=&#8221;https:\/\/higeacbd.com\/wp-content\/uploads\/2020\/10\/Farmacodinamia-y-Farmacocine\u0301tica.jpg&#8221; background_blend=&#8221;soft-light&#8221; custom_padding=&#8221;3vw||1vw|||&#8221;][et_pb_row _builder_version=&#8221;3.25&#8243; background_size=&#8221;initial&#8221; background_position=&#8221;top_left&#8221; background_repeat=&#8221;repeat&#8221;][et_pb_column type=&#8221;4_4&#8243; _builder_version=&#8221;3.25&#8243; custom_padding=&#8221;|||&#8221; custom_padding__hover=&#8221;|||&#8221;][et_pb_cta title=&#8221;Pharmacodynamique et pharmacocin\u00e9tique&#8221; _builder_version=&#8221;4.6.6&#8243; header_level=&#8221;h1&#8243; header_font=&#8221;|800|||||||&#8221; header_font_size=&#8221;45px&#8221; header_line_height=&#8221;1.3em&#8221; body_font=&#8221;|800|||||||&#8221; body_text_color=&#8221;#000000&#8243; body_font_size=&#8221;20px&#8221; body_line_height=&#8221;1.6em&#8221; use_background_color=&#8221;off&#8221; custom_button=&#8221;on&#8221; button_text_size=&#8221;14px&#8221; button_text_color=&#8221;#ffffff&#8221; button_bg_color=&#8221;#00a88d&#8221; button_border_width=&#8221;8px&#8221; button_border_color=&#8221;rgba(47,56,84,0)&#8221; button_border_radius=&#8221;60px&#8221; button_letter_spacing=&#8221;1px&#8221; button_font=&#8221;Montserrat|700||on|||||&#8221; button_use_icon=&#8221;off&#8221; background_layout=&#8221;light&#8221; animation_direction=&#8221;bottom&#8221; header_font_size_tablet=&#8221;&#8221; header_font_size_phone=&#8221;30px&#8221; header_font_size_last_edited=&#8221;on|phone&#8221; button_text_color_hover=&#8221;#ffffff&#8221; button_border_radius_hover=&#8221;66px&#8221; button_letter_spacing_hover=&#8221;1px&#8221; button_bg_color_hover=&#8221;rgba(47,56,84,0.9)&#8221; button_text_size__hover_enabled=&#8221;off&#8221; button_one_text_size__hover_enabled=&#8221;off&#8221; button_two_text_size__hover_enabled=&#8221;off&#8221; button_text_color__hover_enabled=&#8221;on&#8221; button_text_color__hover=&#8221;#ffffff&#8221; button_one_text_color__hover_enabled=&#8221;off&#8221; button_two_text_color__hover_enabled=&#8221;off&#8221; button_border_width__hover_enabled=&#8221;off&#8221; button_one_border_width__hover_enabled=&#8221;off&#8221; button_two_border_width__hover_enabled=&#8221;off&#8221; button_border_color__hover_enabled=&#8221;off&#8221; button_one_border_color__hover_enabled=&#8221;off&#8221; button_two_border_color__hover_enabled=&#8221;off&#8221; button_border_radius__hover_enabled=&#8221;on&#8221; button_border_radius__hover=&#8221;66px&#8221; button_one_border_radius__hover_enabled=&#8221;off&#8221; button_two_border_radius__hover_enabled=&#8221;off&#8221; button_letter_spacing__hover_enabled=&#8221;on&#8221; button_letter_spacing__hover=&#8221;1px&#8221; button_one_letter_spacing__hover_enabled=&#8221;off&#8221; button_two_letter_spacing__hover_enabled=&#8221;off&#8221; button_bg_color__hover_enabled=&#8221;on&#8221; button_bg_color__hover=&#8221;rgba(47,56,84,0.9)&#8221; button_one_bg_color__hover_enabled=&#8221;off&#8221; button_two_bg_color__hover_enabled=&#8221;off&#8221;]<\/p>\n<p>La pharmacologie est une branche de la science qui <strong>\u00e9tudie les m\u00e9dicaments et leurs effets sur les \u00eatres vivants<\/strong><\/p>\n<p>[\/et_pb_cta][\/et_pb_column][\/et_pb_row][\/et_pb_section][et_pb_section fb_built=&#8221;1&#8243; admin_label=&#8221;Products&#8221; _builder_version=&#8221;4.5.1&#8243; background_color=&#8221;#f3f3f1&#8243; custom_padding=&#8221;20px||11px||false|false&#8221;][et_pb_row _builder_version=&#8221;4.5.1&#8243; custom_padding=&#8221;8px||17px|||&#8221;][et_pb_column type=&#8221;4_4&#8243; _builder_version=&#8221;4.5.1&#8243; custom_padding=&#8221;|||&#8221; custom_padding__hover=&#8221;|||&#8221;][et_pb_text _builder_version=&#8221;4.6.6&#8243; text_font=&#8221;|500|||||||&#8221; text_text_color=&#8221;#000000&#8243; quote_font=&#8221;||||||||&#8221; header_font=&#8221;||||||||&#8221; header_2_font=&#8221;|800|||||||&#8221; header_2_font_size=&#8221;40px&#8221; header_2_line_height=&#8221;1.4em&#8221; max_width=&#8221;80%&#8221; max_width_tablet=&#8221;90%&#8221; max_width_phone=&#8221;100%&#8221; max_width_last_edited=&#8221;on|tablet&#8221; module_alignment=&#8221;center&#8221; custom_margin=&#8221;||12px|||&#8221;]<\/p>\n<p>Gr\u00e2ce \u00e0 elle, nous cr\u00e9ons les m\u00e9dicaments qui nous aident \u00e0 gu\u00e9rir nos sympt\u00f4mes et nos maladies. Saviez-vous qu\u2019un m\u00e9dicament se compose de deux parties? Le premier est le <strong>m\u00e9dicament qui est la substance active<\/strong> qui agira sur la cible th\u00e9rapeutique. L\u2019autre partie est compos\u00e9e d\u2019excipients qui est tout ce qui entoure le m\u00e9dicament et vous aide \u00e0 voyager \u00e0 travers notre corps jusqu\u2019\u00e0 ce que vous atteignez la cible th\u00e9rapeutique. Un exemple d\u2019excipients sont les capsules solubles contenues dans les m\u00e9dicaments. Ils sont lentement d\u00e9faits dans nos estomacs lib\u00e9rant progressivement la substance active de sorte qu\u2019il est absorb\u00e9 d\u2019une mani\u00e8re optimale.  Gr\u00e2ce \u00e0 elle, nous cr\u00e9ons les m\u00e9dicaments qui nous aident \u00e0 gu\u00e9rir nos sympt\u00f4mes et nos maladies. Saviez-vous qu\u2019un m\u00e9dicament se compose de deux parties? Le premier est le m\u00e9dicament qui est la substance active qui agira sur la cible th\u00e9rapeutique. L\u2019autre partie est compos\u00e9e d\u2019excipients qui est tout ce qui entoure le m\u00e9dicament et vous aide \u00e0 voyager \u00e0 travers notre corps jusqu\u2019\u00e0 ce que vous atteignez la cible th\u00e9rapeutique. Un exemple d\u2019excipients sont les capsules solubles contenues dans les m\u00e9dicaments. Ils se dissolvent lentement dans notre estomac, lib\u00e9rant progressivement le principe actif afin qu&#8217;il soit absorb\u00e9 de mani\u00e8re optimale. <\/p>\n<p>En pharmacologie, avant d\u2019\u00e9tudier le m\u00e9canisme d\u2019action des m\u00e9dicaments, il est tr\u00e8s important de comprendre deux concepts principaux :<\/p>\n<ul>\n<li>Pharmacocin\u00e9tique (PK)<\/li>\n<li>Pharmacodynamique (PD)<\/li>\n<\/ul>\n<p>[\/et_pb_text][\/et_pb_column][\/et_pb_row][et_pb_row admin_label=&#8221;Produits&#8221; _builder_version=&#8221;4.7.7&#8243; _module_preset=&#8221;default&#8221; custom_margin=&#8221;||0px||false|false&#8221; custom_padding=&#8221;0px||0px||false|false&#8221; global_module=&#8221;16824&#8243;][et_pb_column type=&#8221;4_4&#8243; _builder_version=&#8221;4.5.1&#8243; _module_preset=&#8221;default&#8221; background_enable_color=&#8221;off&#8221;][et_pb_shop type=&#8221;best_selling&#8221; posts_number=&#8221;8&#8243; show_pagination=&#8221;on&#8221; module_class=&#8221;custom-shop&#8221; _builder_version=&#8221;4.8.1&#8243; _module_preset=&#8221;default&#8221; title_font=&#8221;|700|||||||&#8221; custom_margin=&#8221;||0px||false|false&#8221; custom_padding=&#8221;0px||0px||false|false&#8221;][\/et_pb_shop][et_pb_signup mailchimp_list=&#8221;higeacbd|5b4d14cf0e&#8221; first_name_field=&#8221;off&#8221; last_name_field=&#8221;off&#8221; title=&#8221;Abonnez-vous et b\u00e9n\u00e9ficiez d\u2019une r\u00e9duction de 10%&#8221; _builder_version=&#8221;4.8.1&#8243; header_level=&#8221;h4&#8243; header_font=&#8221;|800|||||||&#8221; header_text_align=&#8221;center&#8221; header_text_color=&#8221;#000000&#8243; header_font_size=&#8221;35px&#8221; header_line_height=&#8221;1.2em&#8221; use_background_color=&#8221;off&#8221; custom_button=&#8221;on&#8221; button_text_size=&#8221;16px&#8221; button_text_color=&#8221;#00a88d&#8221; button_bg_color=&#8221;rgba(0,0,0,0)&#8221; button_border_width=&#8221;0px&#8221; button_border_radius=&#8221;0px&#8221; button_letter_spacing=&#8221;2px&#8221; button_font=&#8221;|700||on|||||&#8221; button_use_icon=&#8221;off&#8221; button_custom_padding=&#8221;18px|0px|18px|0px|true|true&#8221; button_custom_padding_tablet=&#8221;14px||14px||true|true&#8221; button_custom_padding_phone=&#8221;12px||12px||true|true&#8221; button_custom_padding_last_edited=&#8221;on|phone&#8221; background_layout=&#8221;light&#8221; header_font_size_tablet=&#8221;25px&#8221; header_font_size_phone=&#8221;20px&#8221; header_font_size_last_edited=&#8221;on|desktop&#8221; button_text_size_tablet=&#8221;14px&#8221; button_text_size_phone=&#8221;12px&#8221; button_text_size_last_edited=&#8221;on|phone&#8221; box_shadow_style_button=&#8221;preset4&#8243; box_shadow_horizontal_button=&#8221;0px&#8221; box_shadow_vertical_button=&#8221;2px&#8221; box_shadow_color_button=&#8221;#00a88d&#8221; button_text_color__hover=&#8221;#28221d&#8221; button_text_color__hover_enabled=&#8221;on|hover&#8221; box_shadow_color_button__hover=&#8221;#000000&#8243; box_shadow_color_button__hover_enabled=&#8221;on|desktop&#8221;][\/et_pb_signup][\/et_pb_column][\/et_pb_row][\/et_pb_section][et_pb_section fb_built=&#8221;1&#8243; _builder_version=&#8221;4.5.1&#8243; _module_preset=&#8221;default&#8221; background_color=&#8221;#f3f3f1&#8243; custom_padding=&#8221;14px||27px|||&#8221;][et_pb_row _builder_version=&#8221;4.5.1&#8243; _module_preset=&#8221;default&#8221; custom_padding=&#8221;12px||13px|||&#8221;][et_pb_column type=&#8221;4_4&#8243; _builder_version=&#8221;4.5.1&#8243; _module_preset=&#8221;default&#8221;][et_pb_text _builder_version=&#8221;4.6.6&#8243; _module_preset=&#8221;default&#8221; header_2_font=&#8221;|800|||||||&#8221; header_2_text_align=&#8221;center&#8221; header_2_font_size=&#8221;35px&#8221; header_2_line_height=&#8221;1.2em&#8221; header_3_font=&#8221;|800|||||||&#8221; header_3_text_align=&#8221;center&#8221; max_width=&#8221;80%&#8221; max_width_tablet=&#8221;90%&#8221; max_width_phone=&#8221;100%&#8221; max_width_last_edited=&#8221;on|tablet&#8221; module_alignment=&#8221;center&#8221; custom_margin=&#8221;||-5px|||&#8221; custom_padding=&#8221;||0px|||&#8221;]<\/p>\n<h2>Qu\u2019est-ce que la pharmacocin\u00e9tique?<\/h2>\n<p>Son \u00e9tymologie vient du grec et se r\u00e9f\u00e8re au mouvement des drogues. De fa\u00e7on g\u00e9n\u00e9rale, <strong>la pharmacocin\u00e9tique est ce que l\u2019organisme fait avec les m\u00e9dicaments.<\/strong> D\u00e9crit l\u2019absorption, la distribution, le m\u00e9tabolisme et l\u2019excr\u00e9tion des compos\u00e9s. C\u2019est pourquoi plusieurs fois quand nous allons chez le m\u00e9decin et sont prescrits un m\u00e9dicament toujours nous poser quelques questions qui visent \u00e0 d\u00e9tecter s\u2019il ya un de nos rouages internes qui peuvent affecter la pharmacocin\u00e9tique du m\u00e9dicament que nous allons prendre. Par exemple, si nous avons des probl\u00e8mes de rein, de foie ou de circulation qui interf\u00e9reront avec la circulation normale du m\u00e9dicament \u00e0 travers notre corps.<\/p>\n<p>Par cons\u00e9quent, lorsque nous parlons de pharmacocin\u00e9tique, nous nous concentrons sur l\u2019\u00e9tude de l\u2019entr\u00e9e et la sortie du m\u00e9dicament dans notre corps.<\/p>\n<h3>L\u2019entr\u00e9e:<\/h3>\n<p>Lorsqu\u2019une substance entre, il est important de savoir de quelle fa\u00e7on elle entre et \u00e0 quelle vitesse. Les voies d\u2019administration les plus courantes sont orales et intraveineuses. Apr\u00e8s avoir su dans quelle direction le m\u00e9dicament est entr\u00e9 et \u00e0 quelle vitesse, c\u2019est-\u00e0-dire que nous <a href=\"https:\/\/higeacbd.com\/fr\/datos\/biodisponibilite-et-cbd\" title=\"Biodisponibilit\u00e9 et CBD\">connaissons sa biodisponibilit\u00e9,<\/a>nous pouvons proc\u00e9der \u00e0 l\u2019\u00e9tude de son absorption. L\u2019absorption comprend le processus au cours duquel le compos\u00e9 se d\u00e9place de la voie d\u2019administration au plasma. Comme un dernier processus d\u2019entr\u00e9e, il est important de savoir comment le m\u00e9dicament est distribu\u00e9 \u00e0 travers notre corps.<\/p>\n<h3>La sortie :<\/h3>\n<p>Une fois que le m\u00e9dicament a \u00e9t\u00e9 absorb\u00e9 et distribu\u00e9, nous sommes int\u00e9ress\u00e9s \u00e0 savoir comment il quitte le corps. L\u2019\u00e9limination des compos\u00e9s peut \u00eatre par biotransformation, c\u2019est-\u00e0-dire par le corps qui les transforme ou par excr\u00e9tion.<\/p>\n<p>[\/et_pb_text][\/et_pb_column][\/et_pb_row][\/et_pb_section][et_pb_section fb_built=&#8221;1&#8243; disabled_on=&#8221;off|off|off&#8221; admin_label=&#8221;Features&#8221; _builder_version=&#8221;4.5.1&#8243; background_color=&#8221;#f3f3f1&#8243; custom_padding=&#8221;0px|0px|0px|0px&#8221;][et_pb_row column_structure=&#8221;1_2,1_2&#8243; use_custom_gutter=&#8221;on&#8221; gutter_width=&#8221;1&#8243; make_equal=&#8221;on&#8221; admin_label=&#8221;Ligne CTA&#8221; module_class=&#8221; et_pb_row_fullwidth&#8221; _builder_version=&#8221;4.5.1&#8243; width=&#8221;100%&#8221; width_tablet=&#8221;100%&#8221; width_phone=&#8221;&#8221; width_last_edited=&#8221;on|desktop&#8221; max_width=&#8221;100%&#8221; max_width_tablet=&#8221;100%&#8221; max_width_phone=&#8221;&#8221; max_width_last_edited=&#8221;on|desktop&#8221; custom_padding=&#8221;0px|0px|0px|0px&#8221; make_fullwidth=&#8221;on&#8221;][et_pb_column type=&#8221;1_2&#8243; _builder_version=&#8221;4.5.1&#8243; background_enable_image=&#8221;off&#8221; custom_padding=&#8221;|||&#8221; custom_padding__hover=&#8221;|||&#8221;][et_pb_image src=&#8221;https:\/\/higeacbd.com\/wp-content\/uploads\/2020\/10\/farmacodinamica.jpg&#8221; alt=&#8221;Pharmacodynamie&#8221; title_text=&#8221;Pharmacodynamie&#8221; force_fullwidth=&#8221;on&#8221; _builder_version=&#8221;4.6.6&#8243; _module_preset=&#8221;default&#8221;][\/et_pb_image][\/et_pb_column][et_pb_column type=&#8221;1_2&#8243; _builder_version=&#8221;4.5.1&#8243; background_color=&#8221;#00a88d&#8221; custom_padding=&#8221;|||&#8221; custom_padding__hover=&#8221;|||&#8221;][et_pb_cta title=&#8221;Qu\u2019est-ce que la pharmacodynamique ou la pharmacodynamique?&#8221; button_url=&#8221;#top&#8221; _builder_version=&#8221;4.6.6&#8243; header_font=&#8221;|800|||||||&#8221; header_text_color=&#8221;#ffffff&#8221; body_font=&#8221;Montserrat|500|||||||&#8221; body_text_color=&#8221;#ffffff&#8221; body_link_text_color=&#8221;#000000&#8243; use_background_color=&#8221;off&#8221; custom_button=&#8221;on&#8221; button_text_size=&#8221;16px&#8221; button_text_color=&#8221;#ffffff&#8221; button_bg_color=&#8221;#2f3854&#8243; button_border_width=&#8221;10px&#8221; button_border_color=&#8221;rgba(47,56,84,0)&#8221; button_border_radius=&#8221;60px&#8221; button_letter_spacing=&#8221;1px&#8221; button_font=&#8221;Montserrat|700||on|||||&#8221; button_use_icon=&#8221;off&#8221; button_alignment=&#8221;left&#8221; text_orientation=&#8221;left&#8221; max_width=&#8221;580px&#8221; max_width_tablet=&#8221;&#8221; max_width_phone=&#8221;&#8221; max_width_last_edited=&#8221;on|desktop&#8221; module_alignment=&#8221;left&#8221; custom_margin=&#8221;|||&#8221; custom_padding=&#8221;40px|60px|2px|60px||&#8221; button_text_color_hover=&#8221;#2f3854&#8243; button_border_radius_hover=&#8221;66px&#8221; button_letter_spacing_hover=&#8221;1px&#8221; button_bg_color_hover=&#8221;#ffffff&#8221; button_text_size__hover_enabled=&#8221;off&#8221; button_one_text_size__hover_enabled=&#8221;off&#8221; button_two_text_size__hover_enabled=&#8221;off&#8221; button_text_color__hover_enabled=&#8221;on&#8221; button_text_color__hover=&#8221;#2f3854&#8243; button_one_text_color__hover_enabled=&#8221;off&#8221; button_two_text_color__hover_enabled=&#8221;off&#8221; button_border_width__hover_enabled=&#8221;off&#8221; button_one_border_width__hover_enabled=&#8221;off&#8221; button_two_border_width__hover_enabled=&#8221;off&#8221; button_border_color__hover_enabled=&#8221;off&#8221; button_one_border_color__hover_enabled=&#8221;off&#8221; button_two_border_color__hover_enabled=&#8221;off&#8221; button_border_radius__hover_enabled=&#8221;on&#8221; button_border_radius__hover=&#8221;66px&#8221; button_one_border_radius__hover_enabled=&#8221;off&#8221; button_two_border_radius__hover_enabled=&#8221;off&#8221; button_letter_spacing__hover_enabled=&#8221;on&#8221; button_letter_spacing__hover=&#8221;1px&#8221; button_one_letter_spacing__hover_enabled=&#8221;off&#8221; button_two_letter_spacing__hover_enabled=&#8221;off&#8221; button_bg_color__hover_enabled=&#8221;on&#8221; button_bg_color__hover=&#8221;#ffffff&#8221; button_one_bg_color__hover_enabled=&#8221;off&#8221; button_two_bg_color__hover_enabled=&#8221;off&#8221;]<\/p>\n<p>Pour son \u00e9tymologie aussi grec se r\u00e9f\u00e8re \u00e0 la puissance des m\u00e9dicaments. C\u2019est-\u00e0-dire, l\u2019\u00e9tude de <strong>ce que le m\u00e9dicament fait \u00e0 notre corps.<\/strong> Une fois que le m\u00e9dicament atteint la cible th\u00e9rapeutique, il devra interagir avec les r\u00e9cepteurs cellulaires pour provoquer un effet sur les cellules.<\/p>\n<p>Chaque individu a une r\u00e9ponse diff\u00e9rente aux m\u00e9dicaments. Cependant, la distribution statistique de la r\u00e9ponse aux m\u00e9dicaments de la population est normale (ou cloche gaussienne). Dans cette distribution, nous trouverons une moyenne au centre du capot, des cas extr\u00eames d\u2019hypor\u00e9activit\u00e9 ou d\u2019hyperr\u00e9activit\u00e9 aux extr\u00e9mit\u00e9s de la courbe et aussi des cas idiosyncrasiques qui sont en dehors de la courbe.<\/p>\n<p><img decoding=\"async\" src=\"https:\/\/higeacbd.com\/wp-content\/uploads\/2020\/10\/tolerancia-farmacodinamica.jpg\" width=\"600\" height=\"368\" alt=\"tol\u00e9rance pharmacodynamique\" class=\"wp-image-13537 aligncenter size-full\" srcset=\"https:\/\/higeacbd.com\/wp-content\/uploads\/2020\/10\/tolerancia-farmacodinamica.jpg 600w, https:\/\/higeacbd.com\/wp-content\/uploads\/2020\/10\/tolerancia-farmacodinamica-480x294.jpg 480w\" sizes=\"(min-width: 0px) and (max-width: 480px) 480px, (min-width: 481px) 600px, 100vw\" \/><\/p>\n<p>[\/et_pb_cta][\/et_pb_column][\/et_pb_row][\/et_pb_section][et_pb_section fb_built=&#8221;1&#8243; _builder_version=&#8221;4.5.1&#8243; _module_preset=&#8221;default&#8221; background_color=&#8221;#f3f3f1&#8243; custom_padding=&#8221;14px||27px|||&#8221;][et_pb_row _builder_version=&#8221;4.5.1&#8243; _module_preset=&#8221;default&#8221; custom_padding=&#8221;12px||13px|||&#8221;][et_pb_column type=&#8221;4_4&#8243; _builder_version=&#8221;4.5.1&#8243; _module_preset=&#8221;default&#8221;][et_pb_text _builder_version=&#8221;4.9.1&#8243; _module_preset=&#8221;default&#8221; header_2_font=&#8221;|800|||||||&#8221; header_2_text_align=&#8221;center&#8221; header_2_font_size=&#8221;35px&#8221; header_2_line_height=&#8221;1.2em&#8221; max_width=&#8221;80%&#8221; max_width_tablet=&#8221;90%&#8221; max_width_phone=&#8221;100%&#8221; max_width_last_edited=&#8221;on|tablet&#8221; module_alignment=&#8221;center&#8221; custom_margin=&#8221;||-5px|||&#8221; custom_padding=&#8221;||0px|||&#8221; hover_enabled=&#8221;0&#8243; sticky_enabled=&#8221;0&#8243;]<\/p>\n<p>En outre, si le m\u00e9dicament <strong>est administr\u00e9 de mani\u00e8re r\u00e9p\u00e9t\u00e9e et qu&#8217;il est n\u00e9cessaire<\/strong> d&#8217;<strong> <a href=\"https:\/\/higeacbd.com\/fr\/datos\/tolerance-de-la-cdb\" title=\"Tolerancia CBD\">augmenter la dose, on dit qu&#8217;il g\u00e9n\u00e8re une tol\u00e9rance<\/a><\/strong>. Plus nous avons \u00e0 augmenter la dose pour obtenir les effets d\u00e9sir\u00e9s le plus tol\u00e9rant et d\u00e9pendant de la drogue devient l\u2019individu.<\/p>\n<p>L\u2019\u00e9tude des <strong>effets secondaires des m\u00e9dicaments correspond<\/strong> \u00e0 la branche de la pharmacodynamique. M\u00eame si les effets secondaires ne sont pas ind\u00e9sirables, il est crucial de les conna\u00eetre. Par exemple, si nous voulons conduire, il est pr\u00e9f\u00e9rable de ne pas prendre des antihistaminiques qui ont un effet de somnolence. Celui-ci ne serait pas d\u00e9favorable si au lieu de conduire, nous voulons nous endormir la nuit.<\/p>\n<p>[\/et_pb_text][\/et_pb_column][\/et_pb_row][\/et_pb_section][et_pb_section fb_built=&#8221;1&#8243; admin_label=&#8221;Feature&#8221; _builder_version=&#8221;4.5.1&#8243; background_color=&#8221;#f3f3f1&#8243; background_enable_image=&#8221;off&#8221; custom_padding=&#8221;40px||40px|||&#8221; locked=&#8221;off&#8221;][et_pb_row column_structure=&#8221;2_5,3_5&#8243; _builder_version=&#8221;4.4.4&#8243; locked=&#8221;off&#8221;][et_pb_column type=&#8221;2_5&#8243; _builder_version=&#8221;4.4.4&#8243;][et_pb_image src=&#8221;https:\/\/higeacbd.com\/wp-content\/uploads\/2020\/07\/cbd-aceite-comprar.jpg&#8221; alt=&#8221;tol\u00e9rance pharmacodynamique&#8221; title_text=&#8221;tol\u00e9rance pharmacodynamique&#8221; _builder_version=&#8221;4.6.6&#8243; _module_preset=&#8221;default&#8221;][\/et_pb_image][\/et_pb_column][et_pb_column type=&#8221;3_5&#8243; _builder_version=&#8221;4.4.4&#8243; custom_padding_tablet=&#8221;|20%|||false|false&#8221; custom_padding_phone=&#8221;&#8221; custom_padding_last_edited=&#8221;on|tablet&#8221;][et_pb_text _builder_version=&#8221;4.6.6&#8243; header_2_font=&#8221;|800|||||||&#8221; header_2_text_color=&#8221;#000000&#8243; header_2_font_size=&#8221;40px&#8221; header_2_line_height=&#8221;1.2em&#8221; custom_margin=&#8221;||||false|false&#8221; custom_margin_tablet=&#8221;|||0%|false|false&#8221; custom_margin_last_edited=&#8221;off|desktop&#8221; header_2_font_size_tablet=&#8221;35px&#8221; header_2_font_size_phone=&#8221;25px&#8221; header_2_font_size_last_edited=&#8221;on|phone&#8221;]<\/p>\n<h2>Tol\u00e9rance pharmacodynamique<\/h2>\n<p>[\/et_pb_text][et_pb_text _builder_version=&#8221;4.6.6&#8243; text_font_size_tablet=&#8221;14px&#8221; text_font_size_last_edited=&#8221;off|desktop&#8221; locked=&#8221;off&#8221;]<\/p>\n<p>La pharmacodynamique \u00e9tudie \u00e9galement <strong>les interactions m\u00e9dicamenteuses.<\/strong> Il existe des relations de synergie dans lesquelles les effets d\u2019un ou des deux m\u00e9dicaments augmentent ou s\u2019am\u00e9liorent. L\u2019effet de facilitation des m\u00e9dicaments est \u00e9galement largement utilis\u00e9 en pharmacologie. Dans ces cas, les effets de l\u2019un des m\u00e9dicaments facilitent l\u2019action de l\u2019autre. Par exemple, l\u2019acide clabulamique est utilis\u00e9 en conjonction avec la p\u00e9nicilline pour emp\u00eacher les bact\u00e9ries de g\u00e9n\u00e9rer une r\u00e9sistance aux antibiotiques.<\/p>\n<p>L\u2019\u00e9tude de la dose en pharmacodynamique est importante pour d\u00e9terminer <strong>les marges th\u00e9rapeutiques et d\u2019innocuit\u00e9 de chaque m\u00e9dicament,<\/strong>pour savoir \u00e0 partir de quelle dose le m\u00e9dicament aura un effet sur l\u2019individu et \u00e0 partir de quelle dose il peut \u00eatre mortel. Gr\u00e2ce aux courbes de dose &#8211; r\u00e9ponse, nous pouvons savoir comment chaque dose se comporte.<\/p>\n<p>[\/et_pb_text][\/et_pb_column][\/et_pb_row][\/et_pb_section][et_pb_section fb_built=&#8221;1&#8243; disabled_on=&#8221;off|off|off&#8221; admin_label=&#8221;Features&#8221; _builder_version=&#8221;4.5.1&#8243; background_color=&#8221;#f3f3f1&#8243; custom_padding=&#8221;0px|0px|0px|0px&#8221;][et_pb_row column_structure=&#8221;1_2,1_2&#8243; use_custom_gutter=&#8221;on&#8221; gutter_width=&#8221;1&#8243; make_equal=&#8221;on&#8221; admin_label=&#8221;Ligne CTA&#8221; module_class=&#8221; et_pb_row_fullwidth&#8221; _builder_version=&#8221;4.5.1&#8243; width=&#8221;100%&#8221; width_tablet=&#8221;100%&#8221; width_phone=&#8221;&#8221; width_last_edited=&#8221;on|desktop&#8221; max_width=&#8221;100%&#8221; max_width_tablet=&#8221;100%&#8221; max_width_phone=&#8221;&#8221; max_width_last_edited=&#8221;on|desktop&#8221; custom_padding=&#8221;0px|0px|0px|0px&#8221; make_fullwidth=&#8221;on&#8221;][et_pb_column type=&#8221;1_2&#8243; _builder_version=&#8221;4.5.1&#8243; background_enable_image=&#8221;off&#8221; custom_padding=&#8221;|||&#8221; custom_padding__hover=&#8221;|||&#8221;][et_pb_image src=&#8221;https:\/\/higeacbd.com\/wp-content\/uploads\/2020\/10\/interaccion-farmacodinamica.jpg&#8221; alt=&#8221;interaction pharmacodynamique&#8221; title_text=&#8221;interaction pharmacodynamique&#8221; force_fullwidth=&#8221;on&#8221; _builder_version=&#8221;4.6.6&#8243; _module_preset=&#8221;default&#8221;][\/et_pb_image][\/et_pb_column][et_pb_column type=&#8221;1_2&#8243; _builder_version=&#8221;4.5.1&#8243; background_color=&#8221;#00a88d&#8221; custom_padding=&#8221;|||&#8221; custom_padding__hover=&#8221;|||&#8221;][et_pb_cta title=&#8221;Interaction pharmacodynamique&#8221; button_url=&#8221;#top&#8221; _builder_version=&#8221;4.6.6&#8243; header_font=&#8221;|800|||||||&#8221; header_text_color=&#8221;#ffffff&#8221; body_font=&#8221;Montserrat|500|||||||&#8221; body_text_color=&#8221;#ffffff&#8221; body_link_text_color=&#8221;#000000&#8243; use_background_color=&#8221;off&#8221; custom_button=&#8221;on&#8221; button_text_size=&#8221;16px&#8221; button_text_color=&#8221;#ffffff&#8221; button_bg_color=&#8221;#2f3854&#8243; button_border_width=&#8221;10px&#8221; button_border_color=&#8221;rgba(47,56,84,0)&#8221; button_border_radius=&#8221;60px&#8221; button_letter_spacing=&#8221;1px&#8221; button_font=&#8221;Montserrat|700||on|||||&#8221; button_use_icon=&#8221;off&#8221; button_alignment=&#8221;left&#8221; text_orientation=&#8221;left&#8221; max_width=&#8221;580px&#8221; max_width_tablet=&#8221;&#8221; max_width_phone=&#8221;&#8221; max_width_last_edited=&#8221;on|desktop&#8221; module_alignment=&#8221;left&#8221; custom_margin=&#8221;|||&#8221; custom_padding=&#8221;40px|60px|2px|60px||&#8221; button_text_color_hover=&#8221;#2f3854&#8243; button_border_radius_hover=&#8221;66px&#8221; button_letter_spacing_hover=&#8221;1px&#8221; button_bg_color_hover=&#8221;#ffffff&#8221; button_text_size__hover_enabled=&#8221;off&#8221; button_one_text_size__hover_enabled=&#8221;off&#8221; button_two_text_size__hover_enabled=&#8221;off&#8221; button_text_color__hover_enabled=&#8221;on&#8221; button_text_color__hover=&#8221;#2f3854&#8243; button_one_text_color__hover_enabled=&#8221;off&#8221; button_two_text_color__hover_enabled=&#8221;off&#8221; button_border_width__hover_enabled=&#8221;off&#8221; button_one_border_width__hover_enabled=&#8221;off&#8221; button_two_border_width__hover_enabled=&#8221;off&#8221; button_border_color__hover_enabled=&#8221;off&#8221; button_one_border_color__hover_enabled=&#8221;off&#8221; button_two_border_color__hover_enabled=&#8221;off&#8221; button_border_radius__hover_enabled=&#8221;on&#8221; button_border_radius__hover=&#8221;66px&#8221; button_one_border_radius__hover_enabled=&#8221;off&#8221; button_two_border_radius__hover_enabled=&#8221;off&#8221; button_letter_spacing__hover_enabled=&#8221;on&#8221; button_letter_spacing__hover=&#8221;1px&#8221; button_one_letter_spacing__hover_enabled=&#8221;off&#8221; button_two_letter_spacing__hover_enabled=&#8221;off&#8221; button_bg_color__hover_enabled=&#8221;on&#8221; button_bg_color__hover=&#8221;#ffffff&#8221; button_one_bg_color__hover_enabled=&#8221;off&#8221; button_two_bg_color__hover_enabled=&#8221;off&#8221;]<\/p>\n<p>La pharmacodynamique comprend \u00e9galement <strong>l\u2019analyse des m\u00e9canismes par lesquels les m\u00e9dicaments agissent dans notre corps.<\/strong> Les m\u00e9dicaments peuvent agir sur des mol\u00e9cules cibles telles que des prot\u00e9ines (enzymes, canaux ioniques, mol\u00e9cules de transport ou r\u00e9cepteurs); L\u2019ADN ; ou des articulations silencieuses (prot\u00e9ines plasmatiques ou liaison sp\u00e9cifique). En outre, il existe des m\u00e9dicaments qui n\u2019agissent pas sur les mol\u00e9cules cibles. Par exemple, lorsque nous ressentons de l\u2019acidit\u00e9 et prenons un antiacide, il n\u2019agira pas sur une mol\u00e9cule cible, mais changera directement le PH de notre estomac pour neutraliser les acides.<\/p>\n<p>Les <strong>interactions les plus courantes en pharmacodynamique sont avec les r\u00e9cepteurs.<\/strong> Ce sont des macromol\u00e9cules qui re\u00e7oivent des stimuli et les transmettent aux cellules pour g\u00e9n\u00e9rer un effet. Les drogues peuvent agir de fa\u00e7on s\u00e9lective pour modifier une fonction sp\u00e9cifique de la cellule o\u00f9 elles agissent. En pharmacologie, l\u2019analogie de la serrure (le r\u00e9cepteur) et de la cl\u00e9 (le m\u00e9dicament) est largement utilis\u00e9e. Si le ligando est agoniste, cela signifie que la serrure ouvrira la porte aux hormones ou aux neurotransmetteurs. S\u2019il est antagoniste, il agira en fermant et en verrouillant la porte.<\/p>\n<p>[\/et_pb_cta][\/et_pb_column][\/et_pb_row][\/et_pb_section][et_pb_section fb_built=&#8221;1&#8243; admin_label=&#8221;Feature&#8221; _builder_version=&#8221;4.5.1&#8243; background_color=&#8221;#f3f3f1&#8243; background_enable_image=&#8221;off&#8221; custom_padding=&#8221;21px||18px|||&#8221; locked=&#8221;off&#8221;][et_pb_row column_structure=&#8221;2_5,3_5&#8243; _builder_version=&#8221;4.5.1&#8243; custom_margin=&#8221;|auto|-2px|auto||&#8221; locked=&#8221;off&#8221;][et_pb_column type=&#8221;2_5&#8243; _builder_version=&#8221;4.5.1&#8243;][et_pb_image src=&#8221;https:\/\/higeacbd.com\/wp-content\/uploads\/2020\/07\/cual-es-el-mejor-aceite-de-cbd.jpg&#8221; alt=&#8221;pharmacodynamique et pharmacocin\u00e9tique&#8221; title_text=&#8221;pharmacodynamique et pharmacocin\u00e9tique&#8221; align=&#8221;center&#8221; _builder_version=&#8221;4.6.6&#8243; background_enable_image=&#8221;off&#8221; background_size=&#8221;contain&#8221; max_width_phone=&#8221;300px&#8221; max_width_last_edited=&#8221;off|tablet&#8221; custom_margin=&#8221;|||-30%|false|false&#8221; custom_margin_tablet=&#8221;|||-15%|false|false&#8221; custom_margin_phone=&#8221;|||-10%|false|false&#8221; custom_margin_last_edited=&#8221;on|phone&#8221; locked=&#8221;off&#8221;][\/et_pb_image][\/et_pb_column][et_pb_column type=&#8221;3_5&#8243; _builder_version=&#8221;4.4.4&#8243; custom_padding_tablet=&#8221;|20%|||false|false&#8221; custom_padding_phone=&#8221;&#8221; custom_padding_last_edited=&#8221;on|tablet&#8221;][et_pb_text _builder_version=&#8221;4.6.6&#8243; text_font_size_tablet=&#8221;14px&#8221; text_font_size_last_edited=&#8221;off|desktop&#8221; locked=&#8221;off&#8221;]<\/p>\n<p>Selon le type de lien chimique entre le r\u00e9cepteur et le ligando (le m\u00e9dicament), il y aura des effets passagers ou plus durables. Plus la liaison (p. ex. un pont Van der Waal) est faible, plus l\u2019effet du m\u00e9dicament sera transitoire. Toutefois, si les articulations de type covalent se produisent (non communes), elles sont des liens permanents avec des changements cellulaires irr\u00e9versibles. Dans ce cas, le r\u00e9cepteur serait inutilis\u00e9 pour la vie et forcer le corps \u00e0 produire un nouveau r\u00e9cepteur.<\/p>\n<p>Lors de l\u2019introduction d\u2019un m\u00e9dicament ou d\u2019une substance dans notre corps, il est essentiel de savoir comment notre corps va le traiter (pharmacocin\u00e9tique) et aussi quels effets il aura sur notre corps (pharmacodynamique). Bien que l\u2019\u00e9tude de population se termine dans une distribution normale, chaque individu est un monde et c\u2019est pourquoi nos caract\u00e9ristiques idiosyncrasiques peuvent affecter le dosage que nous devrions prendre pour atteindre les effets secondaires les moins ind\u00e9sirables et la plus grande efficacit\u00e9 th\u00e9rapeutique.  <strong>Il doit s\u2019agir d\u2019un sp\u00e9cialiste qui examine votre cas et prescrit la dose et les m\u00e9dicaments n\u00e9cessaires pour vous traiter.<\/strong><\/p>\n<p>[\/et_pb_text][\/et_pb_column][\/et_pb_row][\/et_pb_section][et_pb_section fb_built=&#8221;1&#8243; admin_label=&#8221;Art\u00edculos relacionados blog&#8221; _builder_version=&#8221;4.7.0&#8243; background_color=&#8221;#f3f3f1&#8243; background_enable_image=&#8221;off&#8221; custom_padding=&#8221;21px||9px|||&#8221; locked=&#8221;off&#8221;][et_pb_row _builder_version=&#8221;4.5.1&#8243; custom_margin=&#8221;|auto|-2px|auto||&#8221; custom_padding=&#8221;11px||7px|||&#8221; 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En utilisant ce site, vous acceptez de suivre la Politique de confidentialit\u00e9 et toutes les Conditions g\u00e9n\u00e9rales imprim\u00e9es sur ce site.<\/p>\n<p>[\/et_pb_text][\/et_pb_column][\/et_pb_row][\/et_pb_section]<\/p>\n<span class=\"et_bloom_bottom_trigger\"><\/span>","protected":false},"excerpt":{"rendered":"<p>La pharmacodynamique \u00e9tudie l\u2019effet des m\u00e9dicaments sur les \u00eatres vivants. Nous expliquons la pharmacodynamique de l\u2019huile de CBD. 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